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The Peptide Effect
phase 2Skin & Anti-Aging

GHK-Cu

Also known as: Copper Peptide GHK-Cu, Glycyl-L-histidyl-L-lysine:copper(II), Loren Pickart Copper Peptide

GHK-Cu is a naturally occurring copper-binding tripeptide found in human plasma, saliva, and urine. It declines significantly with age, dropping from ~200 ng/mL at age 20 to ~80 ng/mL by age 60. Research shows it activates stem cells, promotes collagen synthesis, reduces inflammation, and may reset gene expression toward a healthier, more youthful pattern.

Key Facts

Mechanism
GHK-Cu delivers bioavailable copper to tissues while activating multiple regenerative pathways. It upregulates collagen I, III, and elastin synthesis via TGF-β signaling, stimulates glycosaminoglycan production, activates metalloproteinases for tissue remodeling, and modulates over 4,000 human genes — suppressing pro-inflammatory (IL-6, TNF-α) and promoting anti-inflammatory and repair genes.
Research Status
phase 2
Half-Life
~12 hours (topical persistence varies)
Molecular Formula
C₁₄H₂₃CuN₆O₄
Primary Use
Skin & Anti-Aging

Benefits

  • Stimulates collagen and elastin production for skin firmness and elasticitystrong
  • Accelerates wound healing and reduces scarringstrong
  • Anti-aging effects — reduces fine lines, wrinkles, and age spotsmoderate
  • Promotes hair growth and increases hair follicle sizemoderate
  • Anti-inflammatory — reduces oxidative damage and free radical productionstrong
  • May modulate gene expression toward a healthier pattern (4,000+ genes)preliminary
  • Supports bone density and joint health via collagen synthesispreliminary

Dosage Protocols

RouteDosage RangeFrequencyNotes
Topical (serum/cream)1–2% concentration1–2× dailyMost common for skin rejuvenation; apply to clean skin
Subcutaneous injection1–2 mgDaily for 10–20 day cyclesFor systemic anti-aging and healing effects
Microneedling (transdermal)1–2% solutionEvery 2–4 weeksCombined with microneedling for enhanced skin penetration

Medical disclaimer

Dosage information is provided for educational reference only. Always follow your prescriber's instructions and consult a qualified healthcare provider before starting any peptide protocol.

Side Effects

  • Skin irritation or redness at application site (topical)common
  • Injection site bruising or swellingcommon
  • Mild nausea (subcutaneous injection)rare
  • Headacherare

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Frequently Asked Questions

What is GHK-Cu and where does it come from?
GHK-Cu (glycyl-L-histidyl-L-lysine:copper) is a naturally occurring tripeptide in human blood plasma. It was first identified by Dr. Loren Pickart in the 1970s. Your body produces it naturally, but levels decline significantly with age — by about 60% between ages 20 and 60.
Is GHK-Cu better applied topically or injected?
For skin-specific benefits (wrinkles, skin texture, scars), topical application is effective and convenient. For systemic effects (joint health, overall anti-aging, hair growth), subcutaneous injection delivers higher bioavailability. Many users combine both approaches.
How long does GHK-Cu take to show results?
Topical: visible skin texture improvements typically appear within 2–4 weeks, with collagen remodeling continuing over 2–3 months. Injection: anti-aging and healing effects are typically reported within 2–4 weeks of daily injection cycles.
Can GHK-Cu promote hair regrowth?
Research suggests GHK-Cu can increase hair follicle size and stimulate growth. A 2012 study showed it was comparable to minoxidil 5% for increasing hair follicle size. It is most effective for early-stage thinning rather than complete baldness.
Is GHK-Cu safe to use with other skincare ingredients?
GHK-Cu is compatible with most skincare ingredients including hyaluronic acid and ceramides. However, avoid using it simultaneously with strong acids (AHA/BHA at high concentrations) or vitamin C serums, as low pH can reduce copper peptide efficacy.

References

  1. 1
    GHK peptide as a natural modulator of multiple cellular pathways in skin regeneration(2015)PubMed ↗
  2. 2
    GHK-Cu may prevent oxidative stress in skin by regulating copper and modifying expression of numerous antioxidant genes(2012)PubMed ↗
  3. 3
    Tripeptide-copper complex GHK-Cu stimulates matrix metalloproteinases(1999)PubMed ↗
  4. 4
    The human tripeptide GHK-Cu in prevention of oxidative stress and degenerative conditions of aging(2012)PubMed ↗

Last updated: 2026-02-14